{"title":"Peptides biologiquement actifs \\ Bloqueurs de canaux ioniques et toxines","description":"\u003cp\u003ePeptanova propose actuellement 51 \u003cstrong\u003ebloqueurs de canaux ioniques\u003c\/strong\u003e différents, dont dix peptides Conotoxine, qui constituent une famille de peptides dédiée.\u003cbr\u003eLes bloqueurs de canaux ioniques proposés, tels que SNX-482 Code 4363-s, l'ibériotoxine, la margatoxine ou la kurtoxine, sont des peptides fabriqués chimiquement et non isolés d'origine animale ou produits par des techniques recombinantes.\u003c\/p\u003e\n\u003cp\u003eBloqueur de canaux sensibles à l'acide (ASIC3) APETx2\u003cbr\u003eBloqueur de canaux ioniques ASIC-1a, ASIC-2a Mambalgin-1\u003c\/p\u003e\n\u003cp\u003eBloqueur de canaux Na+ neuronal sensible à la tétrodotoxine Huwentoxin-IV HWTX-IV\u003cbr\u003eBloqueur de canaux Ca2+ de type T \/ canaux Na+ \/ canaux K+ ProTX-1 et ProTX-II Inhibiteur des purinorécepteurs P2X3 \u003ca href=\"https:\/\/peptanova.de\/product\/purotoxin-1\/\" title=\"Purotoxin-I\"\u003ePurotoxin-I\u003c\/a\u003e\u003c\/p\u003e\n\u003cp\u003eLes canaux ioniques mécanosensibles (MSC) sont omniprésents des organismes unicellulaires aux organismes multicellulaires et participent à de nombreux processus physiologiques, notamment la sensation tactile et douloureuse, l'équilibre hydrique et salin, le contrôle de la pression artérielle, la régulation du volume cellulaire et le contrôle de la turgescence [Physiol. Rev., \u003cb\u003e81\u003c\/b\u003e, 685 (2001)]. L'analyse des fonctions médiées par ces canaux peut être effectuée en utilisant un \u003cstrong\u003ebloqueur de canaux ioniques\u003c\/strong\u003e spécifique avec une sélectivité élevée pour les canaux particuliers.\u003c\/p\u003e\n\u003cp\u003eLes bloqueurs peptidiques des canaux Ca2+ de type T, canaux Ca2+ voltage-dépendants, sont classés selon la nature de leurs sous-unités α1. Les bloqueurs des canaux calciques de type N (Ca2+) sont des outils puissants pour la recherche et le développement de stratégies analgésiques alternatives. Les canaux activés par haute tension (HVA) sont composés de α1A-α1F\/α1S, donnant lieu aux canaux de type L, N, P\/Q et R. Les bloqueurs peptidiques des canaux Ca2+ comme l'Agatoxine, la Calciséptine, la Calcicudine, le SNX-482, la Kurtoxine et l'Agélénine sont spécifiques à chaque canal et peuvent être commandés facilement directement depuis notre stock. PeptaNova propose de nombreux bloqueurs de canaux K+ différents comme la Charybdotoxine, l'Ibériotoxine, la Stichodactyla Toxin ou la Margatoxine.\u003c\/p\u003e\n\u003cp\u003eUne grande variété de bloqueurs de canaux sont disponibles pour une livraison rapide depuis notre magasin de Sandhausen. Tous les articles seront expédiés à température ambiante par service de messagerie et arriveront immédiatement après votre commande. Veuillez visiter les sites suivants pour obtenir plus d'informations sur les peptides bloqueurs de canaux ioniques proposés fabriqués à l'Institut Peptidique.\u003c\/p\u003e","products":[{"product_id":"apamin","title":"Apamine","description":"\u003cp\u003e(Abeille domestique, Apis mellifera)\u003c\/p\u003e","brand":"peptanova","offers":[{"title":"0,5 mg","offer_id":52785938039126,"sku":"4257-V","price":135.0,"currency_code":"EUR","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/1008\/7940\/1302\/files\/4257-v.jpg?v=1777022262"},{"product_id":"omega-conotoxin-mviic","title":"ω-Conotoxine MVIIC","description":"\u003cp\u003e(Escargot de mer, Conus magus)\u003c\/p\u003e","brand":"peptanova","offers":[{"title":"0,1 mg","offer_id":52785944887638,"sku":"4283-S","price":130.0,"currency_code":"EUR","in_stock":true},{"title":"0,5 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